Derivatives of bicyclic amino acids, process for t

专利名称：Derivatives of bicyclic amino acids, process

for their preparation, agents containingthem and their use, as well as bicyclic aminoacids as intermediates, and process forpreparing them

发明人：Urbach, Hansjörg, Dr.,Henning, Rainer,

Dr.,Teetz, Volker, Dr.,Geiger, Rolf, Prof.Dr.,Becker, Reinhard, Dr.,Gaul, Holger

申请号：EP82112007.8申请日：19821224公开号：EP00841A2公开日：19830727

摘要：the invention relates to cis, exo - and trans compounds of the formula i in the n= 0, 1 or 2, r1 = hydrogen, possibly by amino, acylamino or benzoylamino substituiertesalkyl, alkenyl, cycloalkyl, cycloalkenyl, cycloalkylalkyl,aryl or aryl teilhydriertes,

respectively by alkyl, or halogen substituted alkoxy can be, as referred to above in aryi -rest substituiertes aralkyl, a mono - orbicyclischen sulfur or oxygen and \\/ or nitrogenheterocyclenrest or a side chain of a naturally occurring amino acid, r2 = hydrogen, alkyl,alkenyl or aralkyl,y = hydrogen or hydroxy, r = hydrogen or y and z = combined oxygenand x = alkyl, alkenyl, cycloalkyl (c1 - c4), - alkyl (c1 - c4) - alkoxy, hydroxy, halogen, nitro,amino.(c1 - c4) - alkylamino.di - (c1 - c4) alkylamino or methylendioxy mono, di - ortrisubstituiertes aryl, or lndol 3 yl, methods for their manufacturethe containing meansand its use, as well as new bicyclische amino acids as intermediate, and their production.

申请人：HOECHST AKTIENGESELLSCHAFT

地址：65926 Frankfurt am Main DE

国籍：DE

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